List of opioids

This is a list of opioids, opioid antagonists and inverse agonists.

Opium and poppy straw derivatives

Crude opiate extracts whole opium products

  • B&O Supprettes
  • Diascordium
  • Dover's powder
  • Kendal Black Drop
  • Laudanum
  • Mithridate
  • Opium
  • Polish heroin (Compote, Kompot)
  • Paregoric
  • Poppy straw concentrate
  • Poppy tea
  • Smoking opium
  • Theriac

Opium alkaloids

  • Codeine
  • Morphine
  • Oripavine
  • Pseudomorphine
  • Thebaine
Structures
Morphides
Codeine Morphine Oripavine Pseudomorphine Thebaine

Alkaloid salts mixtures

  • Pantopon
  • Papaveretum (Omnopon)
  • Tetrapon

Semisynthetics including Bentley compounds

Morphine family

  • 14-Hydroxymorphine [1]
  • 2,4-Dinitrophenylmorphine
  • 6-Methyldihydromorphine [2]
  • 6-Methylenedihydrodesoxymorphine
  • 6-Acetyldihydromorphine [3]
  • Azidomorphine
  • Chlornaltrexamine
  • Chloroxymorphamine [4]
  • Desomorphine (dihydrodesoxymorphine)
  • Dihydromorphine
  • Ethyldihydromorphine [5]
  • Hydromorphinol
  • Methyldesorphine
  • Morphine methylbromide
  • N-Phenethylnordesomorphine
  • N-Phenethyl-14-ethoxymetopon
  • N-Phenethylnormorphine
  • 6-Nicotinoyldihydromorphine (metabolite of nicodicodeine)
  • RAM-378
  • Ro-1539
Structures of Morphine family
Morphine family
14-Hydroxymorphine 2,4-Dinitrophenylmorphine 6-Methyldihydromorphine 6-Methylenedihydrodesoxymorphine 6-Acetyldihydromorphine hydrochloride
Azidomorphine Chlornaltrexamine Chloroxymorphamine Desomorphine
(Dihydrodesoxymorphine)
Dihydromorphine
Ethyldihydromorphine Hydromorphinol Methyldesorphine N-Phenethylnormorphine 6-nicotinoyldihydromorphine
RAM-378

3,6-diesters of morphine

  • Acetylpropionylmorphine
  • 3,6-Dibutanoylmorphine
  • Diacetyldihydromorphine (dihydroheroin, acetylmorphinol)
  • Dibutyrylmorphine 
  • Dibenzoylmorphine (first designer drug)
  • Diformylmorphine 
  • Dipropanoylmorphine
  • Heroin (diacetylmorphine)
  • Nicomorphine
Structures
3,6-diesters of morphine
Acetylpropionylmorphine 3,6-Dibutanoylmorphine Diacetyldihydromorphine
(dihydroheroin, acetylmorphinol)
Dibutyrylmorphine Dibenzoylmorphine Diformylmorphine
Dipropanoylmorphine Heroin
(diacetylmorphine)
Nicomorphine

Codeine-dionine family

  • 6-Monoacetylcodeine
  • Benzylmorphine
  • Codeine methylbromide
  • Desocodeine 
  • Dimethylmorphine (6-O-Methylcodeine) 
  • Ethyldihydromorphine 
  • Methyldihydromorphine (dihydroheterocodeine)
  • Ethylmorphine (dionine)
  • Heterocodeine
  • Isocodeine 
  • Pholcodine (morpholinylethylmorphine)
  • Myrophine
  • Thebacon
  • Transisocodeine 
Structures
Codeine-dionine family
6-Monoacetylcodeine Benzylmorphine Codeine methylbromide Desocodeine Dimethylmorphine
(6-O-Methylcodeine)
Ethyldihydromorphine Methyldihydromorphine
(dihydroheterocodeine)
Ethylmorphine Heterocodeine Isocodeine
Pholcodine Myrophine Transisocodeine

Morphinones and morphols

  • 14-Cinnamoyloxycodeinone
  • 14-Ethoxymetopon
  • 14-Methoxymetopon
  • 14-Phenylpropoxymetopon
  • 3-Acetyloxymorphone
  • 3,14-Diacetyloxymorphone
  • 7-Spiroindanyloxymorphone
  • 8,14-Dihydroxydihydromorphinone 
  • Acetylcodone 
  • Acetylmorphone
  • α-hydrocodol  (=dihydrocodeine, )
  • Benzhydrocodone
  • Bromoisopropropyldihydromorphinone cas?
  • Codeinone
  • Codoxime
  • Conorfone (codorphone)
  • IBNtxA
  • Thebacon (acetyldihydrocodeinone, dihydrocodeinone enol acetate)
  • Hydrocodone
  • Hydromorphone
  • Hydroxycodeine 
  • Metopon (=methyldihydromorphinone)
  • Morphenol 
  • Morphinone
  • Morphol 
  • N-Phenethyl-14-ethoxymetopon
  • Noroxymorphone
  • Oxycodone
  • Oxymorphol
  • Oxymorphone
  • Pentamorphone
  • Semorphone
Structures
Morphinones and morphols
14-Cinnamoyloxycodeinone 14-Ethoxymetopon 14-Methoxymetopon 14-Phenylpropoxymetopon 7-Spiroindanyloxymorphone
8,14-Dihydroxydihydromorphinone Acetylcodone Acetylmorphone α-hydrocodol
(Dihydrocodeine)
Bromoisopropropyldihydromorphinone
Codeinone Codorphone Codol
(Codeine Phosphate)
Codoxime IBNtxA
Thebacon Hydrocodone Hydromorphone Hydroxycodeine Metopon
(methyldihydromorphinone)
Morphenol Morphinone Morphol N-Phenethyl-14-ethoxymetopon Oxycodone
Oxymorphol Oxymorphone Pentamorphone Semorphone

Morphides

  • α-Chlorocodide (= chlorocodide) 
  • β-Chlorocodide 
  • α-Chloromorphide (= chloromorphide)
  • Bromocodide 
  • Bromomorphide 
  • Chlorodihydrocodide 
  • Chloromorphide
  • Codide 
Structures
Morphides
α-chlorocodide β-chlorocodide Bromomorphide
Chlorodihydrocodide. Chloromorphide Codide

Dihydrocodeine series

  • 14-Hydroxydihydrocodeine
  • Acetyldihydrocodeine
  • Dihydrocodeine
  • Dihydrodesoxycodeine (desocodeine) 
  • Dihydroisocodeine 
  • Nicocodeine
  • Nicodicodeine
Structures
Morphides
14-Hydroxydihydrocodeine Acetyldihydrocodeine Dihydrocodeine Dihydrodesoxycodeine
Dihydroisocodeine Nicocodeine Nicodicodeine

Nitrogen morphine derivatives

  • 1-Nitrocodeine cas?
  • Codeine-N-oxide 
  • Morphine-N-oxide
Structures
Morphides
1-Nitrocodeine Codeine-N-oxide Morphine-N-oxide

Hydrazones

  • Oxymorphazone
Structures
Hydrazones
Oxymorphazone

Halogenated morphine derivatives

  • 1-Bromocodeine 
  • 1-Chlorocodeine 
  • 1-Iodomorphine
Structures
Other open chain opioids

1-Bromocodeine

1-Chlorocodeine

1-Iodomorphine

Active opiate metabolites

  • Codeine-6-glucuronide 
  • Codeine-N-oxide (genocodeine)
  • Heroin-7,8-oxide 
  • Morphine-6-glucuronide
  • 3-Monoacetylmorphine
  • 6-Monoacetylmorphine
  • Morphine-N-oxide (genomorphine)
  • Naltrexol 
  • Norcodeine 
  • Normorphine
Structures
Active opiate metabolites
Codeine-N-oxide Heroin-7,8-oxide Morphine-6-glucuronide 6-Monoacetylmorphine
Morphine-N-oxide Naltrexol Norcodeine Normorphine

Morphinans

Morphinan series

  • 3-Hydroxymorphinan 
  • 4-Chlorophenylpyridomorphinan 
  • Cyclorphan
  • Levargorphan 
  • Levorphanol
  • Levophenacylmorphan
  • Levomethorphan
  • Methorphan (racemethorphan)
  • Morphanol (racemorphanol)
  • Norlevorphanol
  • N-Methylmorphinan 
  • Oxilorphan
  • Phenomorphan
  • Proxorphan
  • Ro4-1539
  • Stephodeline  Xorphanol
Structures
Other morphinans
4-chlorophenylpyridomorphinan Cyclorphan Dextrallorphan Levargorphan Levophenacylmorphan
Levomethorphan Norlevorphanol N-Methylmorphinan Oxilorphan Phenomorphan
Dextromethorphan levomethorphan Morphanol Ro4-1539 Stephodeline Xorphanol

Others

  • 1-Nitroaknadinine * 14-episinomenine 
  • 5,6-Dihydronorsalutaridine 
  • 6-Keto Nalbuphine 
  • Aknadinine 
  • Butorphanol
  • Cephakicine 
  • Cephasamine 
  • Cyprodime
  • Drotebanol
  • Fenfangjine G 
  • Ketorfanol
  • Nalbuphine
  • Nalbuphone
  • Tannagine
Structures
Other Morphinans
1-Nitroaknadinine 14-episinomenine 5,6-Dihydronorsalutaridine 6-Keto Nalbuphine Aknadinine
Butorphanol Cephakicine Cephasamine Cyprodime Drotebanol
Fenfangjine G Nalbuphine Sinococuline Sinomenine Tannagine

Benzomorphans

  • 5,9 alpha-diethyl-2-hydroxybenzomorphan (5,9-DEHB) 
  • 8-Carboxamidocyclazocine (8-CAC)
  • Alazocine
  • Anazocine 
  • Bremazocine
  • Butinazocine 
  • Carbazocine 
  • Cogazocine
  • Cyclazocine
  • Dezocine
  • Eptazocine
  • Etazocine 
  • Ethylketazocine 
  • Fedotozine 
  • Fluorophen 
  • Gemazocine 
  • Ibazocine 
  • Ketazocine
  • Metazocine
  • Moxazocine 
  • Pentazocine
  • Phenazocine
  • Quadazocine 
  • SKF-10047

-->

  • Tonazocine
  • Volazocine
  • Zenazocine
Structures
Benzomorphans
5,9 alpha-diethyl-2-hydroxybenzomorphan
(5,9-DEHB)
8-Carboxamidocyclazocine Alazocine Anazocine Bremazocine
Butinazocine Carbazocine Cogazocine Cyclazocine Dezocine
Eptazocine Etazocine Ethylketocyclazocine Fedotozine Fluorophen
Gemazocine Ibazocine Ketazocine Metazocine Moxazocine
Pentazocine Phenazocine Quadazocine Thiazocine Tonazocine
Volazocine Zenazocine

4-Phenylpiperidines

Pethidines (meperidines)

  • 4-Fluoropethidine
  • Allylnorpethidine
  • Anileridine
  • Benzethidine
  • Carperidine
  • Difenoxin
  • Diphenoxylate
  • Etoxeridine (carbetidine)
  • Furethidine
  • Hydroxypethidine (bemidone)
  • Morpheridine
  • Meperidine-N-oxide 
  • Oxpheneridine (carbamethidine)
  • Pethidine (meperidine)
  • Pethidine intermediate A
  • Pethidine intermediate B (norpethidine)
  • Pethidine intermediate C (pethidinic acid)
  • Pheneridine
  • Phenoperidine
  • Piminodine
  • Properidine (ipropethidine)
  • Sameridine
Structures
Pethidines (meperidines)
4-Fluoropethidine 8-Carboxamidocyclazocine Allylnorpethidine Anileridine Benzethidine
Carperidine Difenoxin Diphenoxylate Etoxeridine Furethidine
Hydroxypethidine Morpheridine Meperidine-N-oxide Oxpheneridine Pethidine
Pethidine intermediate A Pethidine intermediate B Pethidine intermediate C Pheneridine Phenoperidine
Piminodine Properidine Sameridine

Prodines

  • Allylprodine
  • (α/β)-Meprodine
  • Desmethylprodine (MPPP)
  • PEPAP
  • (α/β)-Prodine
  • Prosidol
  • Trimeperidine (promedol)
Structures
Prodines
Allylprodine (α/β)-Meprodine Desmethylprodine (MPPP) PEPAP Prodine
Prosidol Prosidol

Ketobemidones

  • Acetoxyketobemidone
  • Droxypropine
  • Ketobemidone
  • Methylketobemidone
  • Propylketobemidone
Structures
Ketobemidones
Acetoxyketobemidone Droxypropine Ketobemidone Methylketobemidone Propylketobemidone

Others

  • Alvimopan
  • Loperamide
  • LS-115509
  • Picenadol
Structures
Other phenylpiperidines
Alvimopan Loperamide LS-115509 Picenadol

Open chain opioids

Amidones

  • Dextromethadone 
  • Dipipanone
  • Isomethadone=
  • Levoisomethadone 
  • Levomethadone 
  • Methadone
  • Methadone intermediate 
  • Normethadone
  • Norpipanone 
  • Phenadoxone (heptazone)
Structures
Amidones

Dextromethadone

Dipipanone

Isomethadone

Levoisomethadone
Noracetylmethadol Levomethadone Methadone Methadone intermediate
Normethadone Norpipanone Phenadoxone Pipidone

Methadols

  • Acetylmethadol 
  • Alphaacetylmethadol 
  • Alphamethadol 
  • Betacetylmethadol 
  • Betamethadol 
  • Dimepheptanol (racemethadol)
  • Isomethadol 
  • Levacetylmethadol
  • Noracymethadol
Structures
Other open chain opioids

Alphaacetylmethadol

Dimepheptanol

Levacetylmethadol

Noracetylmethadol

Moramides

  • Desmethylmoramide 
  • Dextromoramide
  • Levomoramide
  • Moramide intermediate 
  • Racemoramide
Structures
Other open chain opioids

Desmethylmoramide

Dextromoramide

Levomoramide

Moramide intermediate

Racemoramide

Thiambutenes

  • Diethylthiambutene
  • Dimethylthiambutene
  • Ethylmethylthiambutene
  • Piperidylthiambutene
  • Pyrrolidinylthiambutene
  • Thiambutene
Structures
Thiambutenes

Diethylthiambutene

Dimethylthiambutene

Ethylmethylthiambutene

Piperidylthiambutene

Thiambutene

Tipepidine

Phenalkoxams

  • Dextropropoxyphene (propoxyphene)
  • Dimenoxadol
  • Dioxaphetyl butyrate
  • Levopropoxyphene
  • Norpropoxyphene
  • Pyrroliphene
Structures
Phenalkoxams

Dextropropoxyphene
(propoxyphene)

Dimenoxadol

Dioxaphetyl butyrate

Levopropoxyphene

Norpropoxyphene

Ampromides

  • Diampromide
  • Phenampromide
  • Propiram
Structures
Ampromides

Diampromide

Phenampromide

Propiram

Others

  • Embutramide
  • IC-26
  • Isoaminile
  • Lefetamine
  • R-4066
Structures
Other open chain opioids

Embutramide

IC-26

Isoaminile

Lefetamine

R-4066

Anilidopiperidines

  • 3-Allylfentanyl
  • 3-Methylfentanyl
  • 3-Methylthiofentanyl
  • 4-Phenylfentanyl
  • Alfentanil
  • α-Methylacetylfentanyl
  • α-Methylfentanyl
  • α-Methylthiofentanyl
  • Benzylfentanyl   
  • β-hydroxyfentanyl
  • β-hydroxythiofentanyl
  • β-Methylfentanyl
  • Brifentanil
  • Butyrfentanyl
  • Carfentanil
  • Fentanyl
  • Lofentanil
  • N-Methylcarfentanil
  • Mirfentanil
  • Ocfentanil
  • Ohmefentanyl
  • Parafluorofentanyl
  • Phenaridine
  • R-30490
  • Remifentanil
  • Sufentanil
  • Thenylfentanyl 
  • Thiofentanyl
  • Trefentanil
Structures
Anilidopiperidines
3-Allylfentanyl 3-Methylfentanyl 3-Methylthiofentanyl 4-Phenylfentanyl Alfentanil
Alphamethylacetylfentanyl Alphamethylfentanyl Alphamethylthiofentanyl Benzylfentanyl Betahydroxyfentanyl
Betahydroxythiofentanyl Betamethylfentanyl Brifentanil Carfentanil Fentanyl
Lofentanil Mirfentanil Ocfentanil Ohmefentanyl Parafluorofentanyl
Phenaridine Remifentanil Sufentanil Thenylfentanyl Thiofentanyl
Trefentanil

Oripavine derivatives

  • 7-PET
  • Acetorphine
  • Alletorphine (N-allyl-noretorphine)
  • BU-48
  • Buprenorphine
  • Buprenorphine-3-glucuronide
  • Cyprenorphine
  • Dihydroetorphine
  • Etorphine
  • Homprenorphine
  • 18,19-Dehydrobuprenorphine (HS-599) 
  • N-cyclopropylmethylnoretorphine 
  • Nepenthone 
  • Norbuprenorphine
  • Norbuprenorphine-3-glucuronide
  • Thevinone 
  • Thienorphine
Structures
Oripavine derivatives
7-PET Acetorphine Alletorphine BU-48 Buprenorphine
Cyprenorphine Dihydroetorphine Etorphine Homprenorphine 18,19-Dehydrobuprenorphine
N-cyclopropylmethylnoretorphine Nepenthone Norbuprenorphine Thevinone Thienorphine

Phenazepanes

  • Ethoheptazine
  • Meptazinol
  • Metheptazine
  • Metethoheptazine
  • Proheptazine
Structures
Phenazepanes

Ethoheptazine

Meptazinol

Metheptazine

Metethoheptazine

Proheptazine

Pirinitramides

  • Bezitramide
  • Piritramide
Structures
Pirinitramides

Bezitramide

Piritramide

Benzimidazoles

  • Clonitazene
  • Etonitazene
  • Isotonitazene
  • Metonitazene
Structures
Benzimidazoles

Clonitazene

Etonitazene

Isotonitazene

Metonitazene

Nitazene: R = hydrogen

Indoles

  • 18-Methoxycoronaridine
  • 7-Acetoxymitragynine 
  • 7-Hydroxymitragynine
  • ψ-Akuammigine
  • Akuammidine 
  • Akuammine
  • Coronaridine
  • Eseroline
  • Hodgkinsine
  • Ibogaine
  • Mitragynine
  • Mitragynine pseudoindoxyl
  • Noribogaine
  • Pericine
  • Pseudoakuammigine
Structures
Indoles

18-Methoxycoronaridine

7-Acetoxymitragynine

7-Hydroxymitragynine

Akuammidine

Akuammine

Eseroline

Hodgkinsine

Mitragynine

Pericine

Pseudoakuammigine

Beta-Amino Ketones

  • 3-(dimethylamino)-2,2-dimethyl-1-phenylpropan-1-one
Structures
Indoles

3-(dimethylamino)-2,2-dimethyl-1-phenylpropan-1-one (Beta-amine ketone 'compound 29')

Diphenylmethylpiperazines

  • BW373U86
  • DPI-221
  • DPI-287
  • DPI-3290
  • SNC-80
  • AZD-2327
Structures
Diphenylmethylpiperazines

BW373U86

DPI-221

DPI-287

DPI-3290

SNC-80

Opioid peptides

Dynorphins

  • Big dynorphin
  • Dynorphin A
  • Dynorphin B
  • Leumorphin
Structures
Dynorphins
Big dynorphin Dynorphin A Dynorphin B

Endomorphins

  • Endomorphin-1
  • Endomorphin-2

Endorphins

  • α-Endorphin
  • β-Endorphin
  • γ-Endorphin
  • α-Neoendorphin
  • β-Neoendorphin
Structures
Dynorphins
Beta-endorphin Alpha-endorphin Gamma-endorphin α-neoendorphin β-neoendorphin

Enkephalins

  • DADLE
  • DAMGO
  • Deltorphin 
  • Met-enkephalin
  • Leu-enkephalin
Structures
Enkephalins
DADLE DAMGO Deltorphin Met-enkephalin Leu-enkephalin

Propeptides

  • Proenkephalin
  • Proendorphin
  • Proopiomelanocortin

Others / unknown

  • Adrenorphin
  • Amidorphin
  • Biphalin
  • Casokefamide
  • Casomorphins
  • Cytochrophin-4
  • DALDA (Tyr-D-Arg-Phe-Lys-NH2)
  • Deltorphin I
  • Deltorphin II
  • Deprolorphin
  • Dermorphin
  • DPDPE 
  • Frakefamide
  • Gliadorphin
  • Gluten exorphins
  • Hemorphin-4
  • Metkefamide
  • Morphiceptin
  • Nociceptin
  • Octreotide
  • Opiorphin
  • Rubiscolin
  • Soymorphins
  • Spinorphin
  • TRIMU 5
  • Tynorphin
  • Valorphin
  • Zyklophin
Structures
Other or unknown opioid peptides
Adrenorphin Amidorphin Casomorphin DALDA Deltorphin
Dermorphin DPDPE Endomorphin-1
Endomorphin-2
Gliadorphin Morphiceptin
Nociceptin Octreotide Opiorphin Rubiscolin TRIMU 5

Others

  • 3-(3-Methoxyphenyl)-3-ethoxycarbonyltropane 
  • AD-1211
  • AH-7921
  • Axomadol
  • Azaprocin
  • BDPC
  • Bisnortilidine 
  • BRL-52537
  • Bromadol
  • Bromadoline
  • Ciprefadol
  • Ciramadol
  • Doxpicomine
  • Enadoline
  • Faxeladol
  • GR-89696
  • Herkinorin
  • ICI-199,441
  • ICI-204,448
  • Ketamine
  • KNT-42
  • LPK-26
  • Lufuradom
  • Metofoline
  • MT-45
  • Desmethylclozapine
  • Nexeridine
  • NNC 63-0532
  • Nortilidine
  • O-Desmethyltramadol
  • Phenadone
  • Phencyclidine
  • Prodilidine
  • Profadol
  • Ro64-6198
  • Salvinorin A
  • Salvinorin B ethoxymethyl ether
  • Salvinorin B methoxymethyl ether
  • SB-612,111
  • SC-17599
  • RWJ-394,674
  • TAN-67
  • Tapentadol
  • Thiobromadol (C-8813)
  • Tifluadom
  • Tilidine
  • Tramadol
  • Trimebutine
  • U-47700
  • U-50,488
  • U-69,593
  • Viminol
  • 1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide (W-18)

Opioid antagonists and inverse agonists

  • 4-Caffeoyl-1,5-quinide
  • 5'-Guanidinonaltrindole
  • β-Funaltrexamine
  • 6β-Naltrexol
  • 6β-Naltrexol-d4
  • Alvimopan
  • AT-076
  • Binaltorphimine
  • BU09059
  • Buprenorphine
  • Chlornaltrexamine
  • Clocinnamox
  • Cyclazocine
  • Cyprodime
  • Diacetylnalorphine 
  • Diprenorphine (M5050)
  • Fedotozine
  • ICI-174864
  • J-113,397
  • JDTic
  • JTC-801
  • Levallorphan
  • LY-2456302
  • LY-255582
  • Methocinnamox
  • Methylnaltrexone
  • ML350
  • Naldemedine
  • Nalfurafine
  • Nalmefene
  • Nalmexone
  • Nalodeine (N-allylnorcodeine) 
  • Naloxazone
  • Naloxegol
  • Naloxol
  • Naloxonazine
  • Naloxone
  • Naloxone benzoylhydrazone
  • Nalorphine
  • Naltrexone
  • Naltriben
  • Naltrindole
  • Norbinaltorphimine
  • Oxilorphan
  • PF-4455242
  • S-allyl-3-hydroxy-17-thioniamorphinan (SAHTM)
  • Samidorphan 
  • SR-16430

Biased ligands

  • 6'-Guanidinonaltrindole
  • 7-Hydroxymitragynine
  • Herkinorin
  • ICI-199,441
  • Noribogaine
  • Oliceridine
  • RB-64
  • TRV734

Receptor heteromer targeting ligands

  • 6'-GNTI (δ-κ)
  • CYM-51010 (δ-μ)[6]
  • NNTA (κ-μ)[7]
  • IBNtxA (μ1G-NOP)

Uncategorized opioids

  • ADL-5859
  • Alimadol
  • Amentoflavone
  • Anilopam +HCl
  • Asimadoline
  • Cyproterone acetate
  • FE 200665
  • Fedotozine
  • HZ-2
  • Kolokol-1
  • Matrine
  • MCOPPB
  • Menthol
  • MT-7716
  • Nalfurafine
  • Nalorphine
  • Nalorphine dinicotinate
  • PZM21
  • Proglumide
  • Ro65-6570 
  • SoRI-9409 
  • Spiradoline 
  • SR-8993 
  • SR-16435
Structures
Uncategorized opioids

Alimadol

Anilopam

Asimadoline

FE 200665

Fedotozine

MCOPPB

Nalfurafine

Nalodeine

Nalorphine

Nalorphine dinicotinate

SoRI-9409

Combination drug formulations containing opioids

  • Buprenorphine/naloxone
  • Buprenorphine/samidorphan (ALKS-5461)
  • Co-codamol (codeine phosphate/paracetamol)
  • Co-codaprin (codeine phosphate/aspirin)
  • Co-dydramol (dihydrocodeine tartrate/paracetamol)
  • Co-proxamol (dextropropoxyphene/paracetamol)
  • Fentanyl/fluanisone
  • Hydrocodone/ibuprofen
  • Hydrocodone/paracetamol
  • Loperamide/simethicone
  • Morphine/naltrexone
  • Naltrexone/bupropion
  • Oxycodone/aspirin
  • Oxycodone/naloxone
  • Oxycodone/paracetamol

See also

  • List of opioids by visual 2D molecular skeletal renderings (bundled remotely, click "show" after following link)
  • List of Schedule I drugs (US)
  • Gray death

References

  1. ChemIndex CAS Registry Number 3371-56-0
  2. ChemIndex CAS Registry Number 509-56-8
  3. ChemIndex CAS Registry Number 63715-94-6
  4. NCBI PubChem SID 750205
  5. chembase cbid_346222
  6. Gomes I, Fujita W, Gupta A, Saldanha SA, Saldanha AS, Negri A, Pinello CE, Eberhart C, Roberts E, Filizola M, Hodder P, Devi LA (2013). "Identification of a μ-δ opioid receptor heteromer-biased agonist with antinociceptive activity". Proc. Natl. Acad. Sci. U.S.A. 110 (29): 12072–7. Bibcode:2013PNAS..11012072G. doi:10.1073/pnas.1222044110. PMC 3718106. PMID 23818586.
  7. Yekkirala AS, Lunzer MM, McCurdy CR, Powers MD, Kalyuzhny AE, Roerig SC, Portoghese PS (2011). "N-naphthoyl-beta-naltrexamine (NNTA), a highly selective and potent activator of μ/kappa-opioid heteromers". Proc. Natl. Acad. Sci. U.S.A. 108 (12): 5098–103. Bibcode:2011PNAS..108.5098Y. doi:10.1073/pnas.1016277108. PMC 3064379. PMID 21385944.
  • Carbonate derivatives of 14β-hydroxycodeine "viz., 14β-hydroxy-6-O-(methoxycarbonyl)codeine, 6-O-methoxycarbonyl-14β-(methoxycarbonyloxy)codeine, and 14β-acetoxy-6-O-methoxy-carbonylcodeine, potential substrates for ring C modification in morphinane (sic) alkaloids, were synthesized for the first time." Russian Chemical Bulletin. August 2008, Volume 57, Issue 8, pp 1773–1774. Date: 11 Aug 2009; I. V. Evsikova, S. K. Moiseev, P. V. Petrovskii, V. N. Kalinin. Published in Russian in Izvestiya Akademii Nauk. Seriya Khimicheskaya, No. 8, pp. 1739–1740
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